ANXIETY STATES

 

 

Classification of Anxiety Disorders

 

Anxiety States or Disorders as they are currently known include a group of diseases characterized by mobilization of the fight-flight natural mechanism in the absence of a real danger to life or safety of the person. Thus the body reacts by over-sympathetic activity including fast heart beats,  cold extremities, sweating, tremors, gastric spasm, muscle tension, and hyper-vigilance.

 

·        Phobic disorder

1.      Social phobia

2.      Specific phobia

3.      Simple phobia

4.      Agoraphobia

·        Panic disorder

·        Generalised anxiety disorder

·        Mixed anxiety and  depressive disorder

·        Obsessive compulsive disorder

·        Reactions to severe stress and adjustment disorders

·        Acute stress reaction

·        Post-traumatic stress disorder

·        Anxious (avoidant) personality disorder

·        Other anxiety disorder

 

 

Phobic disorder

 

Under phobic disorder are to be included those conditions of abnormally intense dread in the presence of an object or situation often amounting to panic.

 

Agoraphobia is the commonest phobia. Anxiety is produced by, or in anticipation of, going out alone.   Fear often increases progressively the further the patient is away from home. Anxiety tends to occur in crowded places such as trains, buses, shops, restaurants and cinemas or where the patient may feel trapped eq. lifts or hairdressers.

 

 

Certain key items were identified. 

 

The stimulus (presence of situation causing anxiety)

A response

(tried to avoid that situation)

 

Somatic symptoms and Signs

(hand shaky, weak at the knees. sweating. clammy hands. hot and cold feelings, pallor)

 

The autonomic symptoms

include butterflies in the stomach, heart pounds or flutters. dry mouth, dizziness or faintness, difficulty in getting breath, tightness in the chest. 

 

Specific situations

staying at home alone. going out alone, being in an enclosed space and being in crowds.

 

Personality factors differ in normal controls and those with phobic anxiety states which if persistent can become chronic anxiety states.

 

On the Maudsley Personality Inventory which depicts personality on an introversion/extraversion continuum and this is usually pictured on the horizontal axis whereas rising neuroticism is depicted on the vertical axis.  Normal controls are midway on the introversion/extraversion continuum but low on neuroticism.

 

Patients with generalised anxiety disorder (chronic anxiety) had very high neuroticism scores and were found to be the most introverted of any group.  Patients with phobic disorders were less neurotic and less introverted than those with generalised anxiety disorder.  These personal findings have been supported by other workers.

 

 

Acute stress reaction tends to be short-lived and related to major stress,  occurs  in  those  with  a  stable  pre-morbid personality and generally there is no fami   history.

 

 

 

Post-traumatic stress disorder (PTSD) develops after an acute stress reaction.  It is characterised by insomnia, nightmares and flashbacks, during which the original trauma is relived.  This helps to 'fix' the trauma more firmly in the nervous system. During World War I prolonged stress in the trenches led to exhaustion and 'shell-shock’, which would now be called PTSD. The lessons were well learned in World War II when front-line sedation was extensively employed. This resulted in a diminution of insomnia, nightmares and flashbacks and less PTSD.  Although unfashionable, there is still a place for sedation after very traumatic experiences. This is a good way of diminishing the likelihood of PTSD developing later.

 

Generalised  anxiety  disorder is  persistent  and recurrent. Exacerbations of anxiety are precipitated by minor stress. There is usually an abnormal pre-morbid personality with anxious, histrionic or obsessional features and there  is generally a family history of a similar disorder.

 

Differential Diagnosis of Anxiety Disorders

Alcohol withdrawal

Caffeinism

Amphetamines or other stimulant drugs

Hyperthyroid ism

Partial complex seizures

Hypoglycaemia

Cushing' s syndrome

Cardiac arrhythmias (Paroxysmal tachycardia)

Asthma

 

Genetic loading and  sex difference:

 

Nervous disorder in the family of the patient being treated. 

 

fathers also required treatment in               13% of cases

mothers                                                          28%

brothers/sisters in                                         35%. 

 

 

The mean age of onset is between 20 and 30 years of age.

 

In the National Agoraphobia Survey which consisted of a random sample of 100 cases, agoraphobic sufferers reported factors which made them feel  worse  

 

The most common situation reported by 96% was:

 

"having to queue at shops. etc." followed by:

 

"having a definite appointment"

 

'feeling trapped at hairdressers. etc."

 

"domestic arguments and stress"

 

"increase in distance away from hoine"

 

"thinking about £ny problems"

 

"particular places in the neighbourhood"

 

"cloudy1 depressing weather" 'which was reported by 56%.

 

In the same study the factors 'which made patients feel better included:

 

"when cut1 having a way open for a quickreturn home" (91%)

 

"being accompanied by husband or wife"

 

"sitting near a door in hall. restaurant etc."

 

"focusing my mind on something else"

 

"when out for a walk, taking dog, pram1 etc."

 

"talking problem over with a friend"

 

"talking problem over with my doctor"

 

"being accompanied by a friend"

 

“talking sense to myself" (reassuring myself) (52%)

 

"wearing sunglasses" (36%).

 

Who do agoraphobics consult? 

 

In the National Agoraphobic survey it was found that

 

96% consulted their local doctor

77% a psychiatrist

16% a religious or spiritual healer

9% a non-medical hypnotherapist

3% a psychologist

1% phobic societies

 

The outcome of treatment in this very selected sample is illuminating.

                Treatments                 % Receiving Treatment          % Finding it very helpful

                                                                                                          

a)            Tablets/medicine                       96                                            17

 

b)            Relaxation                                  29                                             18

 

c)            Psychotherapyl

                Psychoanalysis                         28                                             15

 

d)            Behaviour therapy/

                Desensitization                         11                                             31

                Flooding etc.

 

e)            Religion/faith

                Healing                                       13                                             15

 

  f)            Hypnotherapy                            15

 

 

Can depression and anxiety states be differentiated?

 

There is a tremendous overlap between the symptoms of depression and anxiety. In doubtful cases there are some facts which help make the

primary diagnosis.  The problem arises because many people with primary depressive disorders develop panic attacks for the first time in their lives.  As the depression recedes, so the panic attacks diminish.  In cases of primary depression there is generally loss of interest, loss of appetite, loss of libido, retardation and the illness develops later in life.  In primary anxiety states there is initial insomnia (difficulty in going off to sleep), phobias, sexual difficulties especially in men, previous attacks of anxiety and the onset is earlier in life.

 

Most people indulge in alcohol as their first line of self-help.  It is essential to take an accurate history because of the patients  vested interest in disguising their drinking habits from their medical advisers. Alcohol is particularly unhelpful since it potentiates the effects of  benzodiazepines, reduces the plasma levels of tricyclic antidepressants. and produces well-known medical complications.

 

THE TREATMENT OF ANXIETY

 

ANXIOLYTICS

 

The benzodiazepines have been phenomenally successful and in 1977 8.000 tonnes of benzodiazepines were consumed annually in the USA. Since then there has been a considerable decline in the prescribing of these very valuable drugs.  In 1983 there were approximately 30 million prescriptions written for benzodiazepine and hypnotics in the UK.

 

It has been estimated by Professor Lader that 15% of the population in developed countries use tranquillisers at some time each year. He estimates that during the past 25 years over 500 million people world wide have taken benzodiazepines.

 

 

It is therefore legitimate to ask how do benzodiazepines decrease anxiety? This can be summarised as follows:-

 

1)      The discovery of benzodiazepine receptors in the brain.

 

2)     The discovery that benzodiazepines work by enhancing the inhibitory neurotransmitter GABA.

 

3)      Thus it appears that the benzodiazepines, anti-anxiety action may be a result of increasing GABA to quiet brain cell activity.

 

Supporting evidence for the role of benzodiazepines has been determined from animal studies. It was found that a decreased number of benzodiazepine receptors appeared in fearful compared with non-fearful rats and emotional compared with non-emotional mice.    It  could be,  therefore,  that  genetic  transmission determines the number of benzodiazepine receptors in man.   If this theory were correct one could postulate that there are fewer benzodiazepine receptors in anxious compared to non-anxious people

 

Benzodiazepine receptor antagonists have now been developed and it has been shown that if these are given to normal healthy volunteers there are increases in hormonal levels, which generally occur with stress, ie. there is an increase in cortisol growth hormone and prolactin.   After the benzodiazepine receptor antagonist was administered the hormonal changes were associated with feelings of sudden panic, agitation, confusion and impending death.  The classical signs of central and peripheral anxiety were observed.

 

The tricyclics and MAOIs exert an anti-anxiety effect by a completely different mechanism.   They affect noradrenergic, adrenergic and serotonergic neurones, which are found especially in the medullary nuclei.  Physiological arousal is due directly to activation of relevant medullary nuclei which can act independently  of  higher  centres which  are  likely  to  be susceptible to effects of tricyclics and MAOIs but which are relatively immune to the direct effects of benzodiazepines.

 

The reaction to withdrawal of benzodiazepines

 

When a benzodiazepine is acutely withdrawn, three things can happen.  If the drug were totally ineffective, then abrupt withdrawal of it will lead to no increase in symptoms of anxiety. This is the neutral reaction.  Because benzodiazepines have long-lasting effects1 when they are withdrawn, there can be a pharmacological withdrawal. Reaction with a peak of symptoms of anxiety at day 14.  If the drug was having no long-term clinical therapeutic benefit, after the pharmacological effect or withdrawing a powerful tranquilliser, the symptoms abate between days 14 and 28 and the patient is no worse off than he was before.

 

 

If the medication had been valuable however, acute withdrawal will lead to rise in symptoms over the following 14 days and a persistent level of symptoms, because the original state of anxiety is no longer being controlled.

 

 

Choice of benzodiazepines

 

 

Table II classifies some of the currently available benzodiazepines according to their elimination half-lives

 

                                                                                                Table II              

Classification of some currently available benzodiazepines accorrding to their elimination half-life­

                Short half-life                     Long half-life

                Alprazolam                        Bromazepam                 Flurazepam

                Lorazepam                        Chlordiazepoxide          Ketazolam

                Loremtazepam                 Clobazam                       Medazepam

                Oxazepam                         Clorazepate                   Nitrazepam

                Temazepam                      Diazepan                        Prazepam

                Triazolam                           Flunitrazepam

 

 

Those with a short half-life are generally good hypnotics because they do not produce as much daytime sedation the following day as benzodiazepines with a long half-life, e.g. temazepam (Normison, Euhypnos).

 

Some studies indicated that triazolam produced more memory disturbance than temazepam.  Largely because of this1 it was withdrawn from the U.K. but is still available in Europe and the USA.  It has a very short half-life and was an excellent hypnotic if getting off to sleep was the major problem.  It was even possible for the medication to be taken at 2 a.m. if patients could not go off to sleep, without leaving much of a hangover.

 

 

Buspirone (Buspar) is thought to reduce the activity of 5HT pathways.  It is unrelated to the benzodiazepines.  It is an Azapirone.  The onset of action is much slower than a benzodiazepine and is an alternative to them. It is ineffective against the rebound anxiety associated with withdrawal of benzodiazepines. It takes 3 weeks to have its full effect and many people withdraw it after 6 weeks.

 

The benzodiazepines with long half-lives can be given as a hypnotic but they will also produce some sedation the following day.  This is often desirable for psychiatric patients.  Chlordiazepoxide (Librium) which is less sedative than diazepam (Valium), clobazam (Frisium) is less sedative than either clorazepate (Tranxene) is becoming more popular, flurazepam (Dalmane and nitrazepam (Nogadon) can lead to quite a lot of sedation the following day.  Flunitrazepam (Rohypnol) has been used in other countries for a long time, but has limited use in Great Britain.

 

 

If an intravenous benzodiazepine is to be used, diazepam can cause problems because the solvent is acid.  This can lead to pain at the site of injection radiating down the arm and it may be followed by venous thrombosis.  A good tip is to withdraw venous into the syringe to dilute the solvent and then inject it slowly back into the vein.  Pain will then not be exper­ienced and the risk of venous thrombosis diminished.  When diazeparn is given for minor surgery or to produce sleep, the best physical sign is to watch the eyelid, as the patient becomes sleepy so the lid will droop. By the time the eyelid has covered half of the pupil most patients will be amnesic from that point onwards. The new intravenous benzodiazepine, midazolam (Hypnovel) is more satisfactory because of its fast onset of recovery and minimal local venous a half-life of two hours and is water soluble compared with diazepam which has an organic solvent. The dose is 2.5 to 7.5 mg. The ampoules are 10 mg in 2 ml.

 

 

It should be recalled that benzodiazepines are powerful muscle relaxants; they should be given with caution to the elderly because big doses can reduce muscle tone. Old ladies are notoriously prone to trip. This can result in the fracture of the neck of the femur and long-acting benzodiazepines can accumulate in the brain. They are best used intermittently or for short courses to reduce the risk of habituation and can be given-2 hours before entering a stressful situation.

 

 

Barbiturates are seldom employed now except for rapid sedation for acute anxiety states. They can also be given as a pre-med prior to ECT. Their ability to produce habituation/addiction, withdrawal fits and to lower the plasma levels of tricyclic antidepressants, are all reasons why their popularity has declined. The major tranquillisers do have a part to play. They can help some chronic anxiety states and they do not produce habituation or addiction and perphenazine (Fentazin) or fluphenazine (Moditen), flupenthixol (Depixol) or trifluoperazine (Stelazine) can all be used in small doses during the day.  If sedation at night is required chlorpromazine (Largactil) can be usefull.

 

Antidepressants can play a valuable part in the treatment of anxiety.  Of the first generation antidepressants clomipramine (Anafranil), imipramine (Tofranil) and dothiepin (Prothiaden) are the ones which are used most commonly.  Dothiepin produces many fewer side-effects than clomipramine.  These drugs can block panic attacks as can monoamine oxidase inhibitors, although one should try the tricyclics initially.  There are some people who do not respond but do extremely well with MAOIs.  Tranylcypromine (Parnate) is the most powerful; phenelzine (Nardil) is highly effective and isocarboxazid (Marplan) can also be valuable.  The incidence of a hypertensive cheese reaction is greatest with tranylcypromine and least with isocarboxazid.  Recent work has demonstrated the safety and efficacy of combined amitriptyline and tranylcypromine.  Indeed it has been demonstrated that amitriptyline will prevent the cheese reaction of monoamine oxidase inhibitors (Pare et al, Lancet, July 24, 1982. p. 183-186).  This work illustrates that it is safer to use combined antidepressants than the MAOI alone. Amitriptyline modifies the rise of blood pressure caused by tyramine.  If certain MAOIs are to be combined with certain tricyclics great care must be taken however. They should be started in small doses simultaneously, giving the sedative tricyclic amitriptyline or trimipramine (Surmontil) at

Might with the.MAOI during the day-morning and lunchtime.  If given later these psychic energisers can induce insomnia.

 

Certain combinations can be lethal; clomipramine (Anafranil) should never be combined with an MAOI; deaths have been reported from this combination.

 

Second Generation antideressants can also be used to treat anxiety states. Trazodone (Molipaxin) is said not to interact with MAOIs. It is sedative and can cause weight loss. Mianserin is also sedative (Bolvidon. Norval). Lofepramine (Gamanil) is a tricyclic with fewer anticholinergic side-effects. On the whole the second generation antidepressants are less effective than the first generation but with the exception of maprotiline (Ludiomil) they are safer if taken in overdosage).

 

The beta-adrenergic blocking drugs have a valuable part to play in the treatment of certain anxiety states. 

 

 

Symptoms of Anxiety

                        Somatic and autonomic                                           Psychic (psychological)

 

                      Palpitations                                                                 Feelings of dread and threat

                      Difficulty in breathing                                                 Irritability

                      Dry mouth                                                                    Panic

                      Nausea                                                                        Anxious anticipation

                      Frequency of micturition                                            Inner (psychic) tension

                      Dizziness                                                                    Worrying over trivia

                      Muscular tension                                                        Difficulty    in concentrating

                      Sweating                                                                     Initial insomnia

                      Abdominal churning                                                   Inability to relax

                      Tremor

                      Cold skin

 

Beta-blockers are best for the treatment of palpitations, tremor, difficulty in breathing, although very occasionally they can precipitate asthma. On the whole they do not influence sweating, gastro-intestinal symptoms, frequency of micturition, nausea or a dry mouth but they can diminish dizziness.  Tremor can be particularly troublesome if it affects a professional musician or a dentist.   Propranolol  (Inderal)  or oxprenolol (Trasicor) 40 mg, given 2 hours before entering a stressful situation is are useful. The dose may occasionally need to be increased to 80-mg.  They can be useful in approximately 10% of anxiety states and their value can be determined very quickly.  Habituation and addiction do not occur.

 

Beta-blockers  can  be  combined,   with  advantage,   with benzodiazepines which are on the whole superior for treating psychic anxiety.  Benzodiazepines should only be used for short courses of treatment.  The benzodiazepines can produce over-sedation whereas small doses of beta adrenergic blocking drugs do not cross the blood-brain barrier and may control tremor, which can be troublesome at interviews and pounding of the heart1 which can be distressing, while leaving intellectual function entirely unimpaired.

 

Benzodiazepines as hypnotics can be given every 3rd night to prevent habituation.

 

Psychological treatments of anxiety

 

individual, group and marital psychotherapy, psychoanalysis, behaviour and cognitive therapy.

Increasing importance is being given to relaxation techniques, the main one being the use of relaxation tapes. 

 

Patients are instructed to use it for 20 minutes twice a day, or if they start to panic or if they have trouble getting to sleep, or wake in the night.

 

biofeedback helps to motivate patients and increases the speed of learning deep muscular relaxation.

 

Other patients prefer yoga or autogenic training.Transcendental Meditation (TM) has been shown to benefit anxiety states, anxiety and alcoholism, mild hypertension, insomnia and stress-related disorders.  Patients are taught to meditate and practise for 20 minutes twice a day.  Studies have shown that regular meditation can decrease anxiety on a number of anxiety scales.  TM can also result in a lower heart rate, blood pressure, respiration rate, basal metabolic rate.  It is also associated with a reduction of alcohol intake, cigarette smoking and the use of minor tranquillisers and hypnotics.  It can also reduce the incidence of hospitalization.   Admissions for heart disease and diseases of the nervous system decreased by 87%, benign and malignant tumours decreased by 55% and mental disorders decreased by 31%.  The most likely explanation for these findings is that the regular use of TM reduces stress. This, in turn, has an effect on the immune system of the body.

 

Other non-drug treatments of anxiety disorders include general reassurance, explanation of symptoms, support, anxiety management and counselling.

 

The role of the therapist

 

It should never be forgotten that the therapist plays an enormous part in the recovery of anxious patients.  There are certain personality types and modes of behaviour, which are helpful.  In a study carried out at Johns Hopkins Hospital, registrars were measured for the three therapeutic virtues of empathy, genuineness and warmth. It was found that registrars possessing these qualities produced a better therapeutic outcome than their psycho-toxic colleagues who were non-empathic, insincere and cold.  Whatever other methods of reducing anxiety are employed; empathy, genuiness and warmth are likely to contribute to the recovery process.